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Facile heterocyclic synthesis and antimicrobial activity of polysubstituted and condensed pyrazolopyranopyrimidine and pyrazolopyranotriazine derivatives


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1. A. B. A. El-Gazzar and H. N. Hafez, Synthesis of 4-substituted pyrido[2,3-d]pyrimidin-4(1H)-one as analgesic and anti-inflammatory agents, Bioorg. Med. Chem. Lett. 19 (2009) 3392-3397; DOI: 10.1016/j.bmcl.2009.05.044.10.1016/j.bmcl.2009.05.044Search in Google Scholar

2. F . M. A. El-Taweel, M. A. Sofan, M. A. Mashaly, M. A. Hanna and A. A. Elagamey, Synthesis of some new pyranoquinoline, pyridine and pyrone derivatives, Pharmazie 45 (1990) 671-673; DOI: 10.1002/chin.199149187.10.1002/chin.199149187Search in Google Scholar

3. A. M. El-Agrody, M. S. Abd El-Latif, N. A. El- Hady, A. H. Fakery and A. H. Bedair, Heteroaromatization with 4-hydroxycoumarin Part II: Synthesis of some new pyrano[2,3-d]-pyrimidines, [1,2,4]triazolo[1,5-c]pyrimidines and pyrimido[1,6-b][1,2,4]triazine derivatives, Molecules 6 (2001) 519-527; DOI: 10.3390/60600519.10.3390/60600519Search in Google Scholar

4. A. H. Bedair, N. A. El-Haddy, M. S. Abd El-Latif, A. H. Fakery and A. M. El-Agrody, 4- Hydroxycoumarin in heterocyclic synthesis. Part III: Synthesis of some new pyrano[2,3-d][1,2,4]triazolo[1,5- c]pyrimidine and pyrimido[1,6-b][1,2,4]triazine derivatives, Farmaco 55 (2000) 708-714; DOI: 10.1016/S0014-827X(00)00097-5.10.1016/S0014-827X(00)00097-5Search in Google Scholar

5. A. M. El-Agrody, M. H. El-Hakim, M. S. Abd El-Latif, A. H. Fakery, E. M. El-sayed and K. A. El- Ghareab, Synthesis of pyrano[2,3-d]pyrimidine and pyrano[3,2-e][1,2,4]triazolo[2,3-c] pyrimidine derivatives with promising antibacterial activities, Acta Pharm. 50 (2000) 111-120.Search in Google Scholar

6. A. G. Martinez and L. J. Marco, Friedlander reaction on 2-amino-3-cyano-4H-pyrans, synthesis of derivatives of 4H-pyran[2,3-b]quinoline, new tacrine analogues, Bioorg. Med. Chem. Lett. 7 (1997) 3165-3170; DOI: 10.1016/S0960-894X(97)10165-2.10.1016/S0960-894X(97)10165-2Search in Google Scholar

7. F . Eiden and F. Denk, Synthesis and CNS activity of pyrane derivatives: 6,8-dioxabicyclo(3,2,1) octanes, Arch. Pharm. (Weinheim) 324 (1991) 353-354.10.1002/ardp.199132406061763946Search in Google Scholar

8. C. P. Dell and C. W. Smith, Antiproliferative derivatives of 4H-naphtho[1,2-b]pyran and process for their preparation, Eur. Pat. 537, 94, 9 21 Apr 1993; ref. Chem. Abstr. 119 (1993) 139102d.Search in Google Scholar

9. F . M. Abdelrazek, P. Metz, N. H. Metwally and S. F. El-Mahrouky, Synthesis and molluscicidal activity of new cinnoline and pyrano[2,3-c]pyrazole derivatives, Arch. Pharm. Chem. Life Sci. 339 (2006) 456-460.10.1002/ardp.20060005716795107Search in Google Scholar

10. G. Bianchi and A. Tava, Synthesis of (2R)(+)-2,3-dihydro-2,6-dimethyl-4H-pyran-4-one, a homologue of pheromones of a species in the hepialidae family, Agr. Biol. Chem. 51 (1987) 2001-2002; DOI: 10.1271/bbb1961.51.2001.10.1271/bbb1961.51.2001Search in Google Scholar

11. K. Noda, A. Nakagawa, Y. Nakajima and H. Ide, Pyrido[2,3-d]-s-triazolo[4,3-c]pyrimidine derivatives, Japan Kokai 7785, 194, 15 Jul 1977; ref. Chem. Abstr. 88 (1978) P50908q.Search in Google Scholar

12. H. N. Hafez, H. A. S. Abbas and A. B. A. El-Gazzar, Synthesis and evaluation of analgesic, antiinflammatory and ulcerogenic activities of some triazolo- and 2-pyrazolyl-pyrido[2,3-d]-pyrimidines, Acta. Pharm. 58 (2008) 359-378; DOI: 10.2478/v10007-008-0024-1.10.2478/v10007-008-0024-119103572Search in Google Scholar

13. A. B. A. El-Gazzar, H. A. R. Hossein and H. N. Hafez, Synthesis and biological evaluation of thieno[2,3-d]pyrimidines derivatives as anti-inflammatory, analgesic and ulcerogenic activity, Acta. Pharm. 57 (2007) 395-411; DOI: 10.2478/v10007-007-0032-6.10.2478/v10007-007-0032-618165185Search in Google Scholar

14. A. B. A. El-Gazzar, H. N. Hafez and G. M. Nawwar, New acyclic nucleosides analogues as potential analgesic, anti-inflammatory, anti-oxidant and anti-microbial derived from pyrimido[4,5-b] quinolines, Eur. Med. Chem. 44 (2009) 1427-1436; DOI: 10.1016/j.ejmech. 2008.09.030.Search in Google Scholar

15. L . P. Prikazchikova, B. M. Khutova, I. F. Vladimirtsev, I. V. Boldyrev and N. I. Zhuravskaya, stimulating activity of mono- and diketone pyrimidine derivatives, Fiziol. Akt. Veshchestva 7 (1975) 84-87; ref. Chem. Abstr. 83 (1975) 127346m.Search in Google Scholar

16. D . J. Brown, Pyrimidines and Their Benzo Derivatives, in Comprehensive Heterocyclic Chemistry (Eds. A. R. Katritzky and C. W. Rees), Vol. 3, Pergamon Press, Oxford 1984, p. 443.10.1016/B978-008096519-2.00035-7Search in Google Scholar

17. S. M. Yu, S. C. Kuo, L. J. Huang, S. S. M. Sun, T. F. Huang and C. M. Teng, Vasorelaxation of rat thoracic aorta caused by two Ca2+-channel blockers, HA-22 and HA-23, J. Pharm. Pharmacol. 44 (1992) 667-671; DOI: 10.1111/j.2042-7158.1992.tb05491.x.10.1111/j.2042-7158.1992.tb05491.xSearch in Google Scholar

18. D . Catarzi, L. Cecchi, V. Colotta, G. Filacchioni, C. Martini, P. Tacchi and A. Lucacchini, Tricyclic heteroaromatic systems. Synthesis and A1 and A2a adenosine binding activities of some 1-aryl-1,4-dihydro-3-methyl[1]benzopyrano[2,3-c]pyrazol-4-ones, 1-aryl-4,9-dihydro-3-methyl-1Hpyrazolo[ 3,4-b]quinolin-4-ones, and 1-aryl-1H-imidazo[4,5-b]quinoxalines, J. Med. Chem. 38 (1995) 1330-1336.10.1021/jm00008a011Search in Google Scholar

19. N . Foloppe, L. M. Fisher, R. Howes, A. Potter, A. G. S. Robertson and A. E. Surgenor, Identification of chemically diverse Chk1 inhibitors by receptor-based virtual screening, Bioorg. Med. Chem. 14 (14) (2006) 4792-4802; DOI: 10.1016/j.bmc.2006.03.021.10.1016/j.bmc.2006.03.021Search in Google Scholar

20. H. M. Al-Matar, K. D. Khalil, A. Y. Adam and M. H. Elnagdi, Green one pot solvent-free synthesis of pyrano[2,3-c]pyrazoles and pyrazolo[1,5-a]pyrimidines, Molecules 15 (2010) 6619-6629; DOI: 10.3390/molecules15096619.10.3390/molecules15096619Search in Google Scholar

21. S. R. Jain and A. Kar, The antibacterial activity of some essential oils and their combination, Planta Med. 20 (1971) 118-123; DOI: 10.1055/s-0028-109967.Search in Google Scholar

22. H. Naeimi, Z. S. Nazifi, S. M. Amininezhad and M. Amouheidari, Synthesis, characterization and in vitro antimicrobial activity of some new Schiff bases and their complexes, J. Antibiot. 66 (2013) 687-689; DOI: 10.1038/ja.2013.73.10.1038/ja.2013.73Search in Google Scholar

23. M . B. Madhusudana Reddy, V. P. Jayashankara and M. A. Pasha, Glycine-catalyzed efficient synthesis of pyranopyrazoles via one-pot multicomponent reaction, Synth. Commun. 40 (2010) 2930-2934; DOI: 10.1080/00397910903340686.10.1080/00397910903340686Search in Google Scholar

24. D . Thomae, G. Kirsch and P. Seck, Synthesis of selenophene analogues of the tacrine series: comparison of classical route and microwave irradiation, Synthesis 10 (2008) 1600-1606; DOI: 10.1055/s-2008-1067001.10.1055/s-2008-1067001Search in Google Scholar

25. N . Galic, B. Peric, B. Kojic-Prodic and Z. Cimerman, Structural and spectroscopic characteristics of aroylhydrazones derived from nicotinic acid hydrazide, J. Mol. Struct. 559 (2001) 187-194; DOI: 10.10.1016/S0022-2860(00)00703-1.10.1016/S0022-2860(00)00703-1Search in Google Scholar

26. V. Klimesova, L. Zahajska, K. Waisser, J. Kaustova and U. Mollmann, Synthesis and antimycobacterial activity of 1, 2, 4-triazole 3-benzylsulfanyl derivatives, Farmaco 59 (2004) 279-288; DOI: 10.1016/j.farmac.2004.01.006. 10.1016/j.farmac.2004.01.00615081345Search in Google Scholar

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