Design and optimization of artemether microparticles for bitter taste masking

T. Yamamoto, T. Nagai, T. Shimura and Y. Yasoshima, Roles of chemical mediators in taste system, Jpn. J. Pharmacol. 76 (1998) 325-348.10.1254/jjp.76.3259623713Search in Google Scholar

P. P. Shah, R. C. Mashru, A. R. Thakkar and A. C. Badhan, Effect of chitosan crosslinking on bitterness evaluation of artemether using response surface methodology, J. Pharm. Pharmacol. 60 (2008) 421-427; DOI: 10.1211/jpp.60.4.0003.10.1211/jpp.60.4.000318380913Search in Google Scholar

P. P. Shah and R. C. Mashru, Development and evaluation of artemether taste masked rapid disintegrating tablets with improved dissolution using solid dispersion technique, AAPS Pharm-SciTech 9 (2008) 494-500; DOI: 10.1208/s12249-008-9066-4.10.1208/s12249-008-9066-4297696118431657Search in Google Scholar

H. Sohi, Y. Sultana and R. K. Khar, Taste masking technologies in oral pharmaceuticals: recent developments and approaches, Drug. Dev. Ind. Pharm. 30 (2004) 429-448; DOI: 10.1081/DDC-120037477.10.1081/DDC-120037477Search in Google Scholar

E. Esposito, R. Rancarati, R. Cortesi, F. Cervellati and C. Nastruzzi, Production of Eudragit microparticles by spray-drying technique: Influence of experimental parameters on morphological and dimensional characteristics, Pharm. Dev. Tech. 5 (2000) 267-278; DOI: 10.1081/PDT-100100541.10.1081/PDT-10010054110810756Search in Google Scholar

Y. Hashimoto, M. Tanaka, H. Kishimoto, H. Shiozawa, K. Hasegawa, K. Matsuyama and T. Uchida, Preparation, characterization and taste masking properties of polyvinylacetal diethylamino acetate microsphere containing trimebutine, J. Pharm. Pharmacol. 54 (2002) 1323-1328.10.1211/00223570276034538312396292Search in Google Scholar

T. Ishikawa, Y. Watanabe, N. Utoguchi and M. Matsumoto, Preparation and evaluation of tablets rapidly disintegrating in saliva containing bitter taste-masked granules by direct compression method, Chem. Pharm. Bull. 47 (1999) 1451-1454.10.1248/cpb.47.145110553641Search in Google Scholar

Y. Gao, F. Cui, Y. Guan, L. Yang, Y. Wang and L. Zhang, Preparation of roxithromycin-polymeric microspheres by the emulsion solvent diffusion method for taste masking, Int. J. Pharm. 318 (2006) 62-69; DOI: 10.1016/j.ijpharm.2006.03.018.10.1016/j.ijpharm.2006.03.01816647230Search in Google Scholar

Y. M. Rane, R. C. Mashru, M. G. Sankalia and J. M. Sankalia, Effect of hydrophilic swellable polymers on dissolution enhancement of carbamazepine solid dispersion studied using response surface methodology, AAPS PharmSciTech 8 (2007) article 27; DOI: 10.1208/pt0802027.10.1208/pt0802027275036717622105Search in Google Scholar

P. P. Shah, R. C. Mashru, Y. M. Rane and A. R. Thakkar, Design and optimization of mefloquine hydrochloride microparticles for bitter taste masking, AAPS PharmSciTech 9 (2008) 377-389; DOI: 10.1208/s12249-008-9052-x.10.1208/s12249-008-9052-x297694418431670Search in Google Scholar

United States Pharmacopoeia XXIV, National Formulary XIX, USP Pharmacopoeilal Convention, Rockville 2000, pp. 1941-1943.Search in Google Scholar

Y. M. Rane, R. C. Mashru, M. G. Sankalia, V. B. Sutariya and P. P. Shah, Investigation on factors affecting chitosan for dissolution enhancement of oxcarbazapine by spray dried microcrystal formulation with an experimental design approach, Drug. Dev. Ind. Pharm. 33 (2007) 1008-1023; DOI: 10.1080/03639040601179749.10.1080/0363904060117974917891588Search in Google Scholar

M. C. Gohel and M. K. Panchal, Novel use of similarity factor f₂ and S_d for the development of diltiazem HCl modified release tablets using a 3² factorial design, Drug. Dev. Ind. Pharm. 28 (2002) 77-87; DOI: 10.1081/DDC-120001488.10.1081/DDC-120001488Search in Google Scholar

T. J. Shah, A. F. Amin, J. R. Parikh and R. H. Parikh, Process optimization and characterization of poloxamer solid dispersion of a poorly water soluble drug, AAPS PharmSciTech 8 (2007) article 29; DOI: 10.1208/pt0802029.10.1208/pt0802029275036917622107Search in Google Scholar

S. Bolton and S. Charles, Pharmaceutical Statistics, Marcel Dekker, New York 2004.Search in Google Scholar

P. M. Satturwar, P. M. Mandaogade and A. K. Dorle, A novel method for preparation of Eudragit RL microcapsules, J. Microencapsul. 19 (2002) 407-413; DOI: 10.1080/02652040210140454.10.1080/0265204021014045412396379Search in Google Scholar

H. Valizadeh, A. Nokhodchi, N. Qarakhani, P. Zakeri-Milani, S. Azarmi, D. Hassanzadeh and R. Lobenberg, Physicochemical characterization of solid dispersions of indomethacin with PEG 6000, Myrj 52, lactose, sorbitol, dextrin and Eudragit E100, Drug. Dev. Ind. Pharm. 30 (2004) 303-317; DOI: 10.1081/DDC-120030426.10.1081/DDC-120030426Search in Google Scholar