Acceso abierto

Synthesis and potential biological activity of some novel 3-[(N-substituted indol-3-yl)methyleneamino]-6-amino-4-aryl-pyrano(2,3-c)pyrazole-5-carbonitriles and 3,6-diamino-4-(N-substituted indol-3-yl)pyrano(2,3-c)pyrazole-5-carbonitriles


Cite

P. Rani, V. K. Srivastava and A. Kumar, Synthesis and anti-inflammatory activity of heterocyclic indole derivatives, Eur. J. Med. Chem. 39 (2004) 449-452; DOI: 10.1016j.egmech2003.11.002.10.1016/j.ejmech.2003.11.002Search in Google Scholar

M. Amir, S. A. Javed and H. Kumar, Synthesis and biological evaluation of some 4-(1H-indol-3-yl)-6-phenyl-1,2,3,4-tetrahydropyrimidin-2-ones/thiones as potent anti-inflammatory agents, Acta Pharm. 58 (2008) 467-477; DOI: 10.2478/v10007-008-0028-x.10.2478/v10007-008-0028-xSearch in Google Scholar

A. H. Mandour, E. R. El-Sawy, K. H. Shaker and M. A. Mustafa, Synthesis, anti-inflammatory, analgesic and anticonvulsant activities of 1,8-dihydro-1-aryl-8-alkyl pyrazolo(3,4-b)indole, Acta Pharm. 60 (2010) 73-88; DOI: 10.2478/v10007-010-0009-8.10.2478/v10007-010-0009-8Search in Google Scholar

N. Siddiqui, M. S. Alam and W. Ahsan, Synthesis, anticonvulsant and toxicity evaluation of 2-(1H-indol-3-yl)acetyl-N-(substituted phenyl) hydrazine carbothioamides and their related heterocyclic derivatives, Acta Pharm. 58 (2008) 445-454; DOI:10.2478/v10007-008-0025-0.10.2478/v10007-008-0025-0Search in Google Scholar

M. A. A. Radwan, E. A. Ragab, N. M. Sabrya and S. M. El-Shenawy, Synthesis and biological evaluation of new 3-substituted indole derivatives as potential anti-inflammatory and analgesic agents, Bioorg. Med. Chem. 15 (2007) 3832-3841; DOI: 10.1016/j.bmc.2007.03.024.10.1016/j.bmc.2007.03.024Search in Google Scholar

E. R. El-Sawy, F. A. Bassyouni, S. H. Abu-Bakr, H. M. Rady and M. M. Abdlla, Synthesis and biological activity of some new 1-benzyl and 1-benzoyl 3-heterocyclic indole derivatives, Acta Pharm. 60 (2010) 55-71; DOI: 10.2478/v10007-010-0004-0.10.2478/v10007-010-0004-0Search in Google Scholar

S. George, M. P. Waran, A. Chakraborty and T. K. Ravi, Synthesis and evaluation of the biological activities of some 3-[5-(6-methyl-4-aryl-2-oxo-1,2,3,4-tetrahydropyrimidin-5-yl)-1,3,4-oxadiazol-2-yl]-imino-1,3-di-hydro-2H-indol-2-one derivatives, Acta Pharm. 58 (2008) 119-129; DOI: 10.2478/v10007-007-0050-4.10.2478/v10007-007-0050-4Search in Google Scholar

M. E. Zaki, H. A. Soliman, O. A. Hiekal and A. E. Z. Rashad, Pyrazolopyranopyrimidines as a class of anti-inflammatory agents, Z. Naturforsch. C 61 (2006) 1-5.10.1515/znc-2006-1-201Search in Google Scholar

S. G. Kuo, L. J. Huang and H. Nakamura, Studies on heterocyclic compounds. 6. Synthesis and analgesic and anti-inflammatory activities of 3,4-dimethylpyrano[2,3-c]pyrazol-6-one derivatives, J. Med. Chem. 27 (1984) 539-544.10.1021/jm00370a020Search in Google Scholar

R. M. Abd El-Aal and M. Younis, Synthesis and antimicrobial activity of certain novel monomethine cyanine dyes, Dyes Pigments 60 (2004) 205-214; DOI: 10.1016/S0143-7208(03)00131-1.10.1016/S0143-7208(03)00131-1Search in Google Scholar

H. M. Al-Matar, K. D. Khalil, A. Y. Adam and M. H. Elnagdi, Green one pot solvent-free synthesis of pyrano[2,3-c]-pyrazoles and pyrazolo[1,5-a]pyrimidines, Molecules 15 (2010) 6619-6629; DOI: 10.3390/molecules15096619.10.3390/molecules15096619625772720877248Search in Google Scholar

A. M. Shestopalov, A. P. Yakubov, D. V. Tsyganov, E. Yanova, M. Yu and V. N. Nesterov, One-pot synthesis of diverse 4-di(tri)fluoromethyl-3-cyanopyridine-2(1H)-thiones and their utilities in the cascade synthesis of annulated heterocycles, Chem. Heterocyc. Compd. 38 (2002) 1180-1189; DOI: 10.1021/cc7001793.10.1021/cc700179318269251Search in Google Scholar

S. Gogoi and C. Zhao, Organocatalyzed enantioselective synthesis of 6-amino-5-cyanodihydropyrano[2,3-c]pyrazole, Tetrahedron Lett. 50 (2009) 2252-2255; DOI: 10.1016/j.tetlet.2009.02.210.10.1016/j.tetlet.2009.02.210274518119915654Search in Google Scholar

A. L. Mndzhoyan, G. L. Papayan, L. D. Zhuruli, S. G. Karagezyan, L. S. Galstyan and V. G. Sarafyan, Synthesis and biological study of hydrazinohydrazones of indole aldehydes and ketons series, Arm. Khim. Zh. (USSR) 22 (1969) 707-713; ref. Chem. Abstr. 72 (1970) 11189f.Search in Google Scholar

A. H. Mandour, E. R. El-Sawy, M. A. Zahran, M. S. Ebaid and M. A. Mustafa, Anti-inflammatory, analgesic, anticonvulsant and antimicrobial activities of some new synthesized N-alkyl-3-indolyl pyrimidines and benzimidazolo(1,2-a) pyrimidines, Biohealth Sci. Bull. (Malaysia) 1 (2009) 57-67.Search in Google Scholar

M. G. Obukowicz, D. J. Welsch, W. J. Salsgiver, M. Berger, K. S. Chinn and K. L. Duffin, Novel, selective delta6 or delta5 fatty acid desaturase inhibitors as anti-inflammatory agents in mice, J. Pharmacol. Exp. Ther. 287 (1998) 157-162.Search in Google Scholar

C. A. Winter, E. A. Risely and G. W. Nuss, Anti-infalmmatory and antipyretic activities of indomethacin, 1-(p-chlorobenzyl)-5-methoxy-2-methyl-indole-3-acetic acid, J. Pharmacol. Exp. Ther. 141 (1963) 369-376.Search in Google Scholar

R. Okun, S. C. Liddon and L. Lasagna, Effect of reserpine pre-treatment on the protective action of amphetamine and phenoxy propazine in the phenylbenzoquinone-induced writhing syndrome in mice, J. Pharm. Exp. Ther. 139 (1963) 107-110; DOI: 10.1038/201306a0.10.1038/201306a014110466Search in Google Scholar

Drug Discovery and Evaluation: Pharmacological Assays, Chapter E: Psychotropic and Neurotropic Activity (Eds. H. G. Vogel and W. H. Vogel, Springer-Verlag), Berlin 1997, pp. 260-261.Search in Google Scholar

A. L. Barry and C. Thornsberry, Susceptibility Testing: Diffusion Test Procedures, in Manual of Clinical Microbiology (Eds. E. H. Lennette, A. Balows, W. J. Hausler, Jr. and J. P. Truant), 3rd ed., American Society for Microbiology, Washington (DC) 1980, pp. 463-474.Search in Google Scholar

eISSN:
1846-9558
ISSN:
1330-0075
Idioma:
Inglés
Calendario de la edición:
4 veces al año
Temas de la revista:
Pharmacy, other