Acceso abierto

Ex vivo permeability study and in vitro solubility characterization of oral Canagliflozin self-nanomicellizing solid dispersion using Soluplus® as a nanocarrier


Cite

Liu X, Zhou L, Zhang F. Reactive melt extrusion to improve the dissolution performance and physical stability of naproxen amorphous solid dispersions. Mol Pharm. 2017;14(3):658–673. Search in Google Scholar

Djuric D, Soluplus. Solubility enhancement with BASF pharma polymers. Reintjes T, editor. BASF SE. 2011; 5:67–72. Search in Google Scholar

Parikh A, Kathawala K, Tan CC, Garg S, Zhou X-F. Self-nanomicellizing solid dispersion of edaravone: part I – oral bioavailability improvement. Drug Des Devel Ther [Internet]. 2018;12:2051–2069. Search in Google Scholar

Hou Y, Wang H, Zhang F, Sun F, Xin M, Li M, et al. Novel self-nanomicellizing solid dispersion based on rebaudioside A: a potential nanoplatforms for oral delivery of curcumin. Int J Nanomedicine [Internet]. 2019;14:557–571. Search in Google Scholar

Younis MA, Tawfeek HM, Abdellatif AAH, Abdel-Aleem JA, Harashima H. Clinical translation of nanomedicines: Challenges, opportunities, and keys. Adv Drug Deliv Rev. 2022;181(114083):114083. Search in Google Scholar

BNF. Pharmaceutical Press is the publishing division of the Royal Pharmaceutical Society. 66-68 East Smithfield, London E1W1AW,UK; 83:2022;769-771. Search in Google Scholar

Singh D, Singh AP, Singh D, Kesavan AK, Arora S, Tiwary AK, et al. Enhanced oral bioavailability and anti-diabetic activity of canagliflozin through a spray dried lipid based oral delivery: a novel paradigm. Daru.2020;28(1):191–208. Search in Google Scholar

Patel NC, Patel HA. A recent solidification approach for nanosuspension: formulation, optimization, and evaluation of canagliflozin immediate release pellets. Folia Med (Plovdiv) [Internet]. 2022;64(3):488–500. Search in Google Scholar

Jassem NA, Abd Alhammid SN. Enhancement of the dissolution and solubility of canagliflozin using nanodispersion systems. Al-Rafidain J Med Sci [Internet]. 2024;6(1):222–31. Search in Google Scholar

Higuchi T, Connors KA. Phase-Solubility Techniques. In: Reilly CN, editor. Advances in Analytical Chemistry and Instrumentation. New York: Wiley-Interscience; 1965. p. 117–212. Search in Google Scholar

Obayes KK, Thomas LM. Development and characterization of hyaluronic acid-incorporated Thermosensitive nasal in situ gel of meclizine hydrochloride. Al-Rafidain J Med Sci [Internet]. 2024;6(1):97–104. Search in Google Scholar

Wang H, He Y, Hou Y, Geng Y, Wu X. Novel self-nanomicellizing formulation based on Rebaudioside A: A potential nanoplatforms for oral delivery of naringenin. Mater Sci Eng C Mater Biol Appl. 2020;112(110926):110926. Search in Google Scholar

Salim FF, A. Rajab N. Formulation and characterization of piroxicam as self-nano emulsifying drug delivery system. Iraqi J Pharm Sci. 2020;29(1):174–183. Search in Google Scholar

Feng S, Zhang Z, Almotairy A, Repka MA. Development and Evaluation of polymeric mixed micelles prepared using hot-melt extrusion for extended delivery of poorly water-soluble drugs. J Pharm Sci . 2023;112(11):2869–2878. Search in Google Scholar

Lu P, Liang Z, Zhang Z, Yang J, Song F, Zhou T, et al. Novel nanomicelle butenafine formulation for ocular drug delivery against fungal keratitis: In Vitro and In Vivo study. Eur J Pharm Sci 2024;192(106629):106629. http://dx.doi.org/10.1016/j.ejps.2023.106629 Search in Google Scholar

Abd allatif K, Hasian JA. Preparation and in vitro evaluation for different types of Ondansetron hydrochloride transdermal patches. Iraqi J Pharm Sci. 2023;32(1):147–155. Search in Google Scholar

Hamed HE, A. Hussein A. Preparation, in vitro and ex-vivo Evaluation of Mirtazapine Nanosuspension and Nanoparticles Incorporated in Orodispersible Tablets. Iraqi J Pharm Sci. 2020;29(1):62–75. Search in Google Scholar

Noor AD, BH. Al-Khedairy E. Formulation and Evaluation of Silymarin Microcrystals by In-Situ Micronization Technique. Iraqi J Pharm Sci. 2019;28(1):1–16. Search in Google Scholar

Singh D, Bedi N, Tiwary AK, Kurmi BD, Bhattacharya S. Natural bio functional lipids containing solid self-micro emulsifying drug delivery system of Canagliflozin for synergistic prevention of type 2 diabetes mellitus. J Drug Deliv Sci Technol 2022;69(103138):103138. Search in Google Scholar

Singh D, Tiwary AK, Bedi N. Role of porous carriers in the biopharmaceutical performance of solid SMEDDS of canagliflozin. Recent Pat Drug Deliv Formul. 2019;12(3):179–98. Search in Google Scholar

Tamer MA, Kassab HJ. The Development of a brain-targeted mucoadhesive amisulpride-loaded nanostructured lipid carrier. Farmacia. 2023;71(5):1032–1044. Search in Google Scholar

Nekkanti V, Wang Z, Betageri GV. Pharmacokinetic Evaluation of Improved Oral Bioavailability of Valsartan: Proliposomes versus self-nanoemulsifying drug delivery system. AAPS PharmSciTech. 2016;17(4):851–862. Search in Google Scholar

Ali SK, Al-Akkam EJM. Oral nanobilosomes of ropinirole: preparation, compatibility and Ex-vivo intestinal absorption study. J Adv Pharm Educ Res. 2023;13(4):8–15. Search in Google Scholar

Jaber SH, Rajab NA. Preparation, in-vitro, ex-vivo, and pharmacokinetic study of lasmiditan as intranasal nanoemulsion-based in situ gel. Pharm Nanotechnol 2024;12. Search in Google Scholar

Zhang X, Li J, Rong R, Wang D, Wang D, Yu Y, et al. Enhancing the oral bioavailability of poorly water-soluble amisupiride with solid nanodispersion. J Drug Deliv Sci Technol. 2023;86(104635):104635. Search in Google Scholar

Pignatello R, Corsaro R, Bonaccorso A, Zingale E, Carbone C, Musumeci T. Soluplus® polymeric nanomicelles improve the solubility of BCS-class II drugs. Drug Deliv Transl Res. 2022;12(8):1991–2006. Search in Google Scholar

Alvarez-Rivera F, Fernández-Villanueva D, Concheiro A, Alvarez-Lorenzo C. Α-lipoic acid in soluplus® polymeric nanomicelles for ocular treating diabetes-associated corneal diseases. J Pharm Sci . 2016;105(9):2855–2863. Search in Google Scholar

Bergonzi MC, Vasarri M, Marroncini G, Barletta E, Degl’Innocenti D. Thymoquinone-loaded soluplus®-Solutol® HS15 mixed micelles: Preparation, in vitro characterization, and effect on the SH-SY5Y cell migration. Molecules. 2020;25(20):4707. Search in Google Scholar

Ha E-S, Baek I-H, Cho W, Hwang S-J, Kim M-S. Preparation and Evaluation of solid dispersion of atorvastatin calcium with Soluplus® by spray drying technique. Chem Pharm Bull (Tokyo). 2014;62(6):545–551. Search in Google Scholar

Sun M, Zhai X, Xue K, Hu L, Yang X, Li G, et al. Intestinal absorption and intestinal lymphatic transport of sirolimus from self-micro emulsifying drug delivery systems assessed using the single-pass intestinal perfusion (SPIP) technique and a chylomicron flow blocking approach: linear correlation with oral bioavailabilities in rats. Eur J Pharm Sci. 2011;43(3):132–140. Search in Google Scholar

Nekkanti V, Wang Z, Betageri GV. Pharmacokinetic Evaluation of Improved Oral Bioavailability of Valsartan: Proliposomes versus self-nanoemulsifying drug delivery system. AAPS Pharm Sci Tech. 2016;17(4):851–862. Search in Google Scholar

eISSN:
2668-7763
Idioma:
Inglés
Calendario de la edición:
6 veces al año
Temas de la revista:
Medicine, Clinical Medicine, other