Open Access

Characterization and taste masking evaluation of microparticles with cetirizine dihydrochloride and methacrylate-based copolymer obtained by spray drying


Cite

1. S. Sharma and S. Lewis, Taste masking technologies: A review, Int. J. Pharm. Pharm. Sci. 2 (2010) 6-13.Search in Google Scholar

2. H. Sohi, Y. Sultana and R. K. Khar, Taste masking technologies in oral pharmaceuticals: recent developments and approaches, Drug Dev. Ind. Pharm. 30 (2004) 429-448; DOI: 10.1081/DDC-120037477.10.1081/DDC-120037477Search in Google Scholar

3. R. Sheshala, N. Khan and Y. Darwis, Formulation and optimization of orally disintegrating tablets of sumatriptan succinate, Chem. Pharm. Bull. 59 (2011) 920-928; DOI: 10.1248/cpb.59.920.10.1248/cpb.59.92021804234Search in Google Scholar

4. R. Matsui, S. Uchida and N. Namiki, Combination effect of physical and gustatory taste masking for propiverine hydrochloride orally disintegrating tablets on palatability, Biol. Pharm. Bull. 38 (2015) 17-22; DOI: 10.1248/bpb.b14-00467.10.1248/bpb.b14-0046725744453Search in Google Scholar

5. Y. D. Yan, J. S. Woo, J. H. Kang, C. S. Yong and H. G. Choi, Preparation and evaluation of tastemasked donepezil hydrochloride orally disintegrating tablets, Biol. Pharm. Bull. 33 (2010) 1364-1370; DOI: 10.1248/bpb.33.1364.10.1248/bpb.33.136420686233Search in Google Scholar

6. D. Douroumis, Practical approaches of taste masking technologies in oral solid forms, Expert Opin. Drug Deliv. 4 (2007) 417-426; DOI: 10.1517/17425247.4.4.417.10.1517/17425247.4.4.41717683254Search in Google Scholar

7. Evonik industries. Products and services: <http://eudragit.evonik.com /product/eudragit/ en/ products-services/eudragit-products/protective-formulations/e-po/Pages/default.aspx>, access date February 24, 2016.Search in Google Scholar

8. M. Szekalska, K. Winnicka, A. Czajkowska-Kośnik, K. Sosnowska and A. Amelian, Evaluation of alginate microspheres with metronidazole obtained by the spray drying technique, Acta Pol. Pharm. Drug Res. 72 (2015) 569-578.Search in Google Scholar

9. D. Guajardo-Flores, C. Rempel, J. A. Gutierrez-Uribe and S. O. Serna-Saldivar, Influence of excipients and spray drying on the physical and chemical properties of nutraceutical capsules containing phytochemicals from black bean extract, Molecules 20 (2015) 21626-21635; DOI: 0.3390/ molecules201219792.10.3390/molecules201219792633207126633352Search in Google Scholar

10. K. Sollohub and K. Cal, Spray drying technique: II Current applications in pharmaceutical technology, J. Pharm. Sci. 99 (2010) 587-597; DOI: 10.1002/jps.21963.10.1002/jps.2196319862804Search in Google Scholar

11. M. Szekalska, A. Amelian and K. Winnicka, Alginate microspheres obtained by the spray drying technique as mucoadhesive carriers of ranitidine, Acta Pharm. 65 (2015) 15-27; DOI: 10.1515/acph-2015-0008.10.1515/acph-2015-000825781701Search in Google Scholar

12. Drug & Drug Target Database. DrugBank version 4.3.: <http://www.drugbank.ca/drugs/DB00341>, access date February 24, 2016.Search in Google Scholar

13. M. Ali, M. A. El-Massik, O. Y. Abdallah and H. Abdelkader, Reduction of bitterness and enhancing palatability of cetirizine oral liquid dosage forms by cyclodextrins, JPDD 2 (2014) 102-110; DOI: 10.15744/2348-9782.1.302.10.15744/2348-9782.1.302Search in Google Scholar

14. R. Mishra and A. Amin, Optimization and characterization of rapidly dissolving films of cetirizine hydrochloride using cyclodextrins for taste masking, Int. J. PharmTech Res. 5 (2013) 536-552.Search in Google Scholar

15. M. Preis, L. Grother, P. Axe and J. Breitkreutz, In-vitro and in-vivo evaluation of taste-masked cetirizine hydrochloride formulated in oral lyophilisates, Int. J. Pharm. 491 (2015) 8-16; DOI: 10.1016/j. ijpharm.2015.06.002.Search in Google Scholar

16. M. Maniruzzaman, M. Bonnefille, A. Aranyos, M. J. Snowden and D. Douroumis, An in vivo and in vitro taste masking evaluation of bitter melt-extruded drugs, J. Pharm. Pharmacol. 66 (2014) 323-337; DOI: 10.1111/jphp.12169.10.1111/jphp.1216924180412Search in Google Scholar

17. D. D. Douroumis, A. Gryczke and S. Schminke, Development and evaluation of cetirizine HCl taste-masked oral disintegrating tablets, AAPS PharmSciTech. 12 (2011) 141-151; DOI: 10.1208/ s12249-010-9569-7.10.1208/s12249-010-9569-7306635521181510Search in Google Scholar

18. D. Douroumis, Orally disintegrating dosage forms and taste-masking technologies, Expert Opin. Drug Deliv. 8 (2011) 665-675; DOI: 10.1517/17425247.2011.566553.10.1517/17425247.2011.56655321438776Search in Google Scholar

19. M. Pein, D. Kirsanov, P. Ciosek, M. Del Valle, I. Yaroshenko, M. Wesoły, M. Zabadaj, A. Gonzalez- Calabuig, W. Wróblewski and A. Legin, Independent comparison study of six different electronic tongues applied for pharmaceutical analysis, J. Pharm. Biomed. Analysis 114 (2015) 321-329; DOI: 10.1016/j.jpba.2015.05.026.10.1016/j.jpba.2015.05.02626099261Search in Google Scholar

20. M. Jańczyk, A. Kutyła, K. Sołłohub, H. Wosicka, K. Cal and P. Ciosek, Electronic tongue for the detection of taste-masking microencapsulation of active pharmaceutical substances, Bioelectrochemistry 80 (2010) 94-98; DOI: 10.1016/j.bioelechem.2010.08.006.10.1016/j.bioelechem.2010.08.00620869333Search in Google Scholar

21. K. Sołłohub, M. Jańczyk, A. Kutyła, H. Wosicka, P. Ciosek and K. Cal, Taste masking of roxithromycin by spray drying technique Acta Pol. Pharm. Drug Res. 68 (2011) 601-604.Search in Google Scholar

22. B. Paw, G. Misztal, H. Hopkała and J. Drozd, Development and validation of a HPLC method for the determination of cetirizine in pharmaceutical dosage forms, Pharmazie 57 (2002) 313-315.Search in Google Scholar

23. A. Jelińska, B. Stanisz, M. Zając, W. Musiał and A. Ostrowicz, Determination of cetirizine dichloride in tablets by HPLC method, Acta Pol. Pharm. Drug Res. 57 (2000) 171-173.Search in Google Scholar

24. N. Yüksel, E. Dinç, F. Onur and T. Baykara, Influence of swelling degree on release of nicardipine hydrochloride from acrylic microspheres prepared by solvent evaporation method, Pharm. Dev. Technol. 3 (1998) 115-121; DOI: 10.3109/10837459809028485. 10.3109/108374598090284859532606Search in Google Scholar

25. M. Wesoły, M. Zabadaj, A. Amelian, K. Winnicka, W. Wróblewski and P. Ciosek, Tasting cetirizine- based microspheres with an electronic tongue, Sens. Actuators B: Chem. (2016) in press; DOI: 10.1016/j.snb.2016.06.14710.1016/j.snb.2016.06.147Search in Google Scholar

26. R. P. Patel, M. P. Patel and A. M. Suthar, Spray drying technology: an overview, Indian J. Sci. Technol. 2 (2009) 44-47; DOI: 10.17485/ijst/2009/v2i10/30719Search in Google Scholar

27. S. Singh and D. Dixit, A review on spray drying: emerging technology in food industry, IJAER, 4 (2014) 1-8.Search in Google Scholar

28. D. E. Dobry, D. M. Settell, J. M. Baumann, R. J. Ray, L. J. Graham and R. A. Beyerinck, A modelbased methodology for spray-drying process development, J. Pharm. Innov. 4 (2009) 133-142; DOI: 10.1007/s12247-009-9064-4.10.1007/s12247-009-9064-4283720920234866Search in Google Scholar

29. P. Sipos, R. Rajkó, K. Pintye-Hódi, I. Erős and P. Szabó-Révész, Formulation optimization of sustained- release ammonio methacrylate copolymer microspheres. Effects of Log P and concentration of polar cosolvents, and role of the drug/copolymer ratio, Pharmaceutics 3 (2011) 830-847; DOI: 10.3390/pharmaceutics3040830.10.3390/pharmaceutics3040830385706024309310Search in Google Scholar

30. R. B. Mane, C. L. Bhingare and M. R. Bhalekar, Preparation and evaluation of carvedilol microsphere by spray drying technique: Effect of process parameters on formulation, IJPQA, 4 (2013) 4-12.Search in Google Scholar

31. N. B. Kulkarni, P. S. Wakte and J. B. Naik, Metformin hydrochloride microparticles for oral controlled release: effect of formulation variables, Int. J. Pharm. Pharm Sci. 5 (2013) 135-144.Search in Google Scholar

32. P. Ciosek, M. Wesoły, M. Zabadaj, J. Lisiecka, K. Sołłohub, K. Cal and W. Wróblewski, Towards flow-through/flow injection electronic tongue for the analysis of pharmaceuticals, Sens. Actuators B 207 (2015) 1087-1094; DOI: 10.1016/j.snb.2014.07.042.10.1016/j.snb.2014.07.042Search in Google Scholar

33. M. Wesoły, X. Cetó, M. Del Valle, P. Ciosek and W. Wróblewski, Quantitative analysis of active pharmaceutical ingredients (APIs) using a potentiometric electronic tongue in a SIA flow system, Electroanalysis 27 (2015) 1-8; DOI: 10.1002/elan.201500407.10.1002/elan.201500407Search in Google Scholar

34. F. Ahmadi-Motamayel, M. T. Goodarzi, S. S. Hendi, H. Abddsamadi and N. Rafiean, Evaluation of salivary flow rate, pH, buffering capacity, calcium and total protein levels in caries free and caries active adolescence, J. Dent. Oral Hyg. 5 (2013) 35-39; DOI: 10.5897/JDOH12.011.Search in Google Scholar

eISSN:
1846-9558
Language:
English
Publication timeframe:
4 times per year
Journal Subjects:
Pharmacy, other